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CB2 receptor agonist 2
CAS No. 1314230-75-5
CB2 receptor agonist 2 ( 4-Quinolone-3-Carboxamide Furan CB2 Agonist; ZINC72105556 )
Catalog No. M27495 CAS No. 1314230-75-5
CB2 receptor agonist 2 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 2MG | 267 | Get Quote |
|
| 5MG | 422 | Get Quote |
|
| 10MG | 618 | Get Quote |
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| 25MG | 972 | Get Quote |
|
| 50MG | 1305 | Get Quote |
|
| 100MG | 1764 | Get Quote |
|
| 200MG | Get Quote | Get Quote |
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| 500MG | Get Quote | Get Quote |
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| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameCB2 receptor agonist 2
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NoteResearch use only, not for human use.
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Brief DescriptionCB2 receptor agonist 2 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.
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DescriptionCB2 receptor agonist 2 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.(In Vitro):CB2 receptor agonist 2 (compound 4g) (1 ?μM; 72 hours) shows low or no cytotoxicity to Hep-G2 cells.(In Vivo):CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is very potent (with maximal effect being reached already at the 1 mg/kg dose) and has antihyperalgesic effects, efficacious also on the first phase of the nocifensive response and strongly reduced by AM630, a CB2-selective antagonist/inverse agonist .
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Synonyms4-Quinolone-3-Carboxamide Furan CB2 Agonist; ZINC72105556
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PathwayGPCR/G Protein
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TargetCannabinoid Receptor
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RecptorTrypanosoma cruzi
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Research Area——
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Indication——
Chemical Information
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CAS Number1314230-75-5
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Formula Weight488.6
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Molecular FormulaC30H36N2O4
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Purity>98% (HPLC)
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Solubility——
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SMILESO=C(NC12CC3CC(CC(C3)C1)C2)C4=CN(C=5C(OC)=CC(=CC5C4=O)C=6OC=CC6)CCCCC
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Souza DCS, et al. Simplified Derivatives of Dibenzylbutyrolactone Lignans from Hydrocotyle bonariensis as Antitrypanosomal Candidates. Chem Biodivers. 2021 Oct;18(10):e2100515.
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